Acylmethanesulfonamides as new acylating agents for primary amines

Silvia Coniglio; Andrea Aramini; M. Candida Cesta; Sandro Colagioia; Roberto Curti; Fabrizio D'Alessandro; Gaetano D'Anniballe; Valerio D'Elia; Giuseppe Nano; Valerie Orlando; Marcello Allegretti

doi:10.1016/j.tetlet.2004.05.073

Acylmethanesulfonamides as new acylating agents for primary amines

Silvia Coniglio^*, Andrea Aramini, M. Candida Cesta, Sandro Colagioia, Roberto Curti, Fabrizio D'Alessandro, Gaetano D'Anniballe, Valerio D'Elia, Giuseppe Nano, Valerie Orlando, Marcello Allegretti

^*Corresponding author for this work

Research output: Contribution to journal › Article › peer-review

9 Scopus citations

Abstract

A new, simple and efficient procedure for the preparation of secondary amides through internal condensation of acylmethanesulfonamides ammonium salts is described. The selective acylation of mixed primary-secondary amines could be an attractive application of the new method.

Original language	English (US)
Pages (from-to)	5375-5378
Number of pages	4
Journal	Tetrahedron Letters
Volume	45
Issue number	28
DOIs	https://doi.org/10.1016/j.tetlet.2004.05.073
State	Published - Jul 5 2004
Externally published	Yes

Keywords

Acylmethanesulfonamides
Condensation reaction
Mixed primary-secondary amine

ASJC Scopus subject areas

Biochemistry
Drug Discovery
Organic Chemistry

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10.1016/j.tetlet.2004.05.073

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title = "Acylmethanesulfonamides as new acylating agents for primary amines",

abstract = "A new, simple and efficient procedure for the preparation of secondary amides through internal condensation of acylmethanesulfonamides ammonium salts is described. The selective acylation of mixed primary-secondary amines could be an attractive application of the new method.",

keywords = "Acylmethanesulfonamides, Condensation reaction, Mixed primary-secondary amine",

author = "Silvia Coniglio and Andrea Aramini and Cesta, {M. Candida} and Sandro Colagioia and Roberto Curti and Fabrizio D'Alessandro and Gaetano D'Anniballe and Valerio D'Elia and Giuseppe Nano and Valerie Orlando and Marcello Allegretti",

year = "2004",

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day = "5",

doi = "10.1016/j.tetlet.2004.05.073",

language = "English (US)",

volume = "45",

pages = "5375--5378",

journal = "Tetrahedron Letters",

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TY - JOUR

T1 - Acylmethanesulfonamides as new acylating agents for primary amines

AU - Coniglio, Silvia

AU - Aramini, Andrea

AU - Cesta, M. Candida

AU - Colagioia, Sandro

AU - Curti, Roberto

AU - D'Alessandro, Fabrizio

AU - D'Anniballe, Gaetano

AU - D'Elia, Valerio

AU - Nano, Giuseppe

AU - Orlando, Valerie

AU - Allegretti, Marcello

PY - 2004/7/5

Y1 - 2004/7/5

N2 - A new, simple and efficient procedure for the preparation of secondary amides through internal condensation of acylmethanesulfonamides ammonium salts is described. The selective acylation of mixed primary-secondary amines could be an attractive application of the new method.

AB - A new, simple and efficient procedure for the preparation of secondary amides through internal condensation of acylmethanesulfonamides ammonium salts is described. The selective acylation of mixed primary-secondary amines could be an attractive application of the new method.

KW - Acylmethanesulfonamides

KW - Condensation reaction

KW - Mixed primary-secondary amine

UR - http://www.scopus.com/inward/record.url?scp=2942691380&partnerID=8YFLogxK

U2 - 10.1016/j.tetlet.2004.05.073

DO - 10.1016/j.tetlet.2004.05.073

M3 - Article

AN - SCOPUS:2942691380

SN - 0040-4039

VL - 45

SP - 5375

EP - 5378

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 28

ER -

Acylmethanesulfonamides as new acylating agents for primary amines

Abstract

Keywords

ASJC Scopus subject areas

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